Molecule Details
InChIKeyOUSYRGFGEKGPNY-UHFFFAOYSA-N
Compound Name9-[3-sulfamoyl-2-(2H-tetrazol-5-yl)-4-(trifluoromethyl)phenyl]-3,9-diazaspiro[5.5]undecane-3-carboximidamide
Canonical SMILESN=C(N)N1CCC2(CC1)CCN(c1ccc(C(F)(F)F)c(S(N)(=O)=O)c1-c1nnn[nH]1)CC2
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL9.07
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q5GN09 vim-1 Klebsiella pneumoniae Pathogen PF00753 9.7 IC50 BindingDB
C7C422 blaNDM-1 Klebsiella pneumoniae Pathogen PF00753 8.8 IC50 ChEMBL;BindingDB
P52699 Serratia marcescens Pathogen PF00753 8.7 IC50 BindingDB