Molecule Details
InChIKeyOUQSBZMPAZAVIV-UHFFFAOYSA-N
Compound NameN1-(6-(5-(pyridin-3-yl)-1H-pyrazolo[3,4-c]pyridin-3-yl)pyridin-2-yl)ethane-1,2-diamine
Canonical SMILESNCCNc1cccc(-c2n[nH]c3cnc(-c4cccnc4)cc23)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL9.24
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q86V86 PIM3 Homo sapiens Human PF00069 9.7 Ki ChEMBL;BindingDB
P11309 PIM1 Homo sapiens Human PF00069 9.5 Ki ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 8.5 Ki ChEMBL;BindingDB