Molecule Details
InChIKeyOUKAHIJIQWSMIH-BMEJSGBISA-N
Canonical SMILESCCN(CC)CC1CN(CC[C@H](CSc2ccccc2)Nc2ccc(S(=O)(=O)NC(=O)c3ccc(N4CCC([C@@H](O)c5ccccc5-c5ccc(Cl)cc5)CC4)cc3)cc2S(=O)(=O)C(F)(F)F)CCO1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL9.35
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P10415 BCL2 Homo sapiens Human PF00452 PF02180 9.4 IC50 ChEMBL;BindingDB
Q07817 BCL2L1 Homo sapiens Human PF00452 PF02180 9.3 IC50 ChEMBL;BindingDB