Molecule Details
InChIKeyOUJGVKJPCLCCKD-SHJPJZKHSA-N
Compound Name(4R,7S,10S,13R,16S,19R)-19-amino-N-[(2S)-1-amino-3-naphthalen-2-yl-1-oxopropan-2-yl]-7,16-dibenzyl-13-[methyl(naphthalene-2-carbonyl)amino]-6,9,12,15,18-pentaoxo-10-[[4-[(propan-2-ylamino)methyl]phenyl]methyl]-1,2-dithia-5,8,11,14,17-pentazacycloicosane-4-carboxamide
Canonical SMILESCC(C)NCc1ccc(C[C@@H]2NC(=O)[C@@H](N(C)C(=O)c3ccc4ccccc4c3)NC(=O)[C@H](Cc3ccccc3)NC(=O)[C@@H](N)CSSC[C@@H](C(=O)N[C@@H](Cc3ccc4ccccc4c3)C(N)=O)NC(=O)[C@H](Cc3ccccc3)NC2=O)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)4
Pfam Stratification Homologous
Avg pChEMBL7.45
SourceChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (4)
Target Gene Organism Category Pfam pChEMBL Type Source
P30872 SSTR1 Homo sapiens Human PF00001 8.9 IC50 ChEMBL
P31391 SSTR4 Homo sapiens Human PF00001 7.2 IC50 ChEMBL
P32745 SSTR3 Homo sapiens Human PF00001 7.0 IC50 ChEMBL
P35346 SSTR5 Homo sapiens Human PF00001 6.7 IC50 ChEMBL