Molecule Details
InChIKeyOUEYXPDIZLXCBG-CMDGGOBGSA-N
Compound Name4-methyl-N-(3-(2-(6-methyl-5-(2-(thiophen-2-yl)acetamido)-1H-indazol-3-yl)vinyl)phenyl)piperazine-1-carboxamide
Canonical SMILESCc1cc2[nH]nc(/C=C/c3cccc(NC(=O)N4CCN(C)CC4)c3)c2cc1NC(=O)Cc1cccs1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.71
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O14965 AURKA Homo sapiens Human PF00069 7.9 IC50 ChEMBL;BindingDB
O75716 STK16 Homo sapiens Human PF00069 7.9 pIC50 TTD_MultiTarget
Q96GD4 AURKB Homo sapiens Human PF00069 7.3 IC50 ChEMBL;BindingDB