Molecule Details
InChIKeyOTYPWJTWIVTSCQ-UHFFFAOYSA-N
Compound NameN-((5-ethyl-2,4,6-trioxo-hexahydropyrimidin-5-yl)methyl)-4-((2-methylquinolin-4-yl)methoxy)benzamide
Canonical SMILESCCC1(CNC(=O)c2ccc(OCc3cc(C)nc4ccccc34)cc2)C(=O)NC(=O)NC1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.69
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P08253 MMP2 Homo sapiens Human PF00040 PF00045 PF00413 6.7 Ki ChEMBL;BindingDB
P39900 MMP12 Homo sapiens Human PF00045 PF00413 PF01471 6.7 Ki ChEMBL;BindingDB