Molecule Details
InChIKeyOTJCUPAITLBALS-UHFFFAOYSA-N
Compound NameN-[[3-[3-(dimethylamino)propoxy]phenyl]methyl]-4-pyridin-4-ylbenzamide
Canonical SMILESCN(C)CCCOc1cccc(CNC(=O)c2ccc(-c3ccncc3)cc2)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.88
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P10635 CYP2D6 Homo sapiens Human PF00067 7.1 IC50 ChEMBL;BindingDB
O75116 ROCK2 Homo sapiens Human PF25346 PF00069 PF08912 7.1 IC50 ChEMBL;BindingDB
Q13464 ROCK1 Homo sapiens Human PF25346 PF00069 PF08912 6.5 IC50 ChEMBL;BindingDB