Molecule Details
InChIKeyOSTVSACFFDGYPT-FUKCDUGKSA-N
Compound NameN-((S)-1-Carbamimidoyl-2-hydroxy-piperidin-3-yl)-2-(2-oxo-3-phenylmethanesulfonylamino-2H-pyridin-1-yl)-acetamide
Canonical SMILESN=C(N)N1CCC[C@H](NC(=O)Cn2cccc(NS(=O)(=O)Cc3ccccc3)c2=O)C1O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.19
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00734 F2 Homo sapiens Human PF00594 PF00051 PF09396 PF00089 9.3 IC50 ChEMBL;BindingDB
P00742 F10 Homo sapiens Human PF00008 PF14670 PF00594 PF00089 7.7 IC50 ChEMBL;BindingDB
P07477 PRSS1 Homo sapiens Human PF00089 7.6 IC50 ChEMBL;BindingDB