Molecule Details
InChIKeyOSQCAWPFHFCVTA-UHFFFAOYSA-N
Compound Name6-(azetidin-3-ylsulfinyl)-3-(4-piperidin-4-ylphenyl)-2-(2H-tetrazol-5-yl)benzenesulfonamide
Canonical SMILESNS(=O)(=O)c1c([S+]([O-])C2CNC2)ccc(-c2ccc(C3CCNCC3)cc2)c1-c1nn[nH]n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.52
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
C7C422 blaNDM-1 Klebsiella pneumoniae Pathogen PF00753 8.7 IC50 ChEMBL;BindingDB
Q9XAY4 blaVIM Pseudomonas aeruginosa Pathogen PF00753 8.7 IC50 BindingDB
P52699 Serratia marcescens Pathogen PF00753 8.2 IC50 BindingDB