Molecule Details
InChIKeyORWZTKJMAQGECS-TVQXRLMPSA-N
Compound Namemethyl 2-[[(1R,2S,6R,14R,15R,19R)-19-[(2R)-2-hydroxypentan-2-yl]-15-methoxy-5-methyl-13-oxa-5-azahexacyclo[13.2.2.12,8.01,6.02,14.012,20]icosa-8(20),9,11,16-tetraen-11-yl]oxymethyl]prop-2-enoate
Canonical SMILESC=C(COc1ccc2c3c1O[C@H]1[C@@]4(OC)C=C[C@@]5(C[C@@H]4[C@](C)(O)CCC)[C@@H](C2)N(C)CC[C@]315)C(=O)OC
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.67
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P41143 OPRD1 Homo sapiens Human PF00001 8.8 IC50 ChEMBL;BindingDB
P35372 OPRM1 Homo sapiens Human PF00001 8.6 IC50 ChEMBL
P41145 OPRK1 Homo sapiens Human PF00001 8.6 IC50 ChEMBL