Molecule Details
InChIKeyORWKFKYYOVHTJR-FOEQRGQYSA-N
Compound Name[(4S,4aS,8aR)-2-[(2S)-2-methyl-3-(2-methyl-1,3-benzoxazol-5-yl)propyl]-3,4,4a,5,6,7,8,8a-octahydro-1H-isoquinolin-4-yl]-[4-(3,4-difluorophenyl)piperazin-1-yl]methanone
Canonical SMILESCc1nc2cc(C[C@H](C)CN3C[C@@H]4CCCC[C@@H]4[C@H](C(=O)N4CCN(c5ccc(F)c(F)c5)CC4)C3)ccc2o1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.43
SourceChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P32745 SSTR3 Homo sapiens Human PF00001 8.5 Kd ChEMBL
P31391 SSTR4 Homo sapiens Human PF00001 6.4 Kd ChEMBL