Molecule Details
InChIKeyORNISAOKGBZAIY-UHFFFAOYSA-N
Canonical SMILESCCOC(=O)C(C)(C)n1nc(-c2cc(-n3c(C)cc(OCc4ncc(F)cc4F)c(Cl)c3=O)c(C)cn2)ccc1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.7
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P28482 MAPK1 Homo sapiens Human PF00069 7.7 IC50 ChEMBL;BindingDB
Q16539 MAPK14 Homo sapiens Human PF00069 7.7 IC50 ChEMBL