Molecule Details
InChIKeyORMLOSONIQIDBI-UHFFFAOYSA-N
Compound Name6-Hydroxy-4-(4-trifluoromethyl-benzylamino)-quinazoline-8-carboxylic acid amide
Canonical SMILESNC(=O)c1cc(O)cc2c(NCc3ccc(C(F)(F)F)cc3)ncnc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.92
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q96GD4 AURKB Homo sapiens Human PF00069 9.6 IC50 ChEMBL;BindingDB
O14965 AURKA Homo sapiens Human PF00069 9.5 IC50 ChEMBL;BindingDB
P23443 RPS6KB1 Homo sapiens Human PF00069 PF00433 7.6 IC50 ChEMBL;BindingDB