Molecule Details
InChIKeyORLPHOALLZATDZ-UHFFFAOYSA-N
Compound NameN-[2-[4-[4-(Trifluoromethoxy)phenoxy]phenylsulfonyl]-1-[(dimethylsulfamoyl)methyl]ethyl]-N-hydroxyformamide
Canonical SMILESCN(C)S(=O)(=O)CC(CS(=O)(=O)c1ccc(Oc2ccc(OC(F)(F)F)cc2)cc1)N(O)C=O
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL9.07
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P08253 MMP2 Homo sapiens Human PF00040 PF00045 PF00413 10.0 pIC50 TTD_MultiTarget
Q9ULZ9 MMP17 Homo sapiens Human PF00045 PF00413 PF01471 9.1 pIC50 TTD_MultiTarget
P14780 MMP9 Homo sapiens Human PF00040 PF00045 PF00413 8.1 IC50 ChEMBL;BindingDB