Molecule Details
InChIKeyOQIIPRFMLCIWTR-QMOZSOIISA-N
Compound Name(4S)-4-[[(2S)-2-[[(2S)-2-[(5-chloro-1H-indole-2-carbonyl)amino]-3-naphthalen-2-ylpropanoyl]amino]-3-(2H-tetrazol-5-yl)propanoyl]amino]-5-oxo-5-[4-(trifluoromethoxy)anilino]pentanoic acid
Canonical SMILESO=C(O)CC[C@H](NC(=O)[C@H](Cc1nn[nH]n1)NC(=O)[C@H](Cc1ccc2ccccc2c1)NC(=O)c1cc2cc(Cl)ccc2[nH]1)C(=O)Nc1ccc(OC(F)(F)F)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.19
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P15884 TCF4 Homo sapiens Human PF00010 6.2 Ki ChEMBL
P35222 CTNNB1 Homo sapiens Human PF00514 6.2 Ki ChEMBL;BindingDB
P36402 TCF7 Homo sapiens Human PF08347 PF00505 6.2 Ki ChEMBL