Molecule Details
InChIKeyOPZCPKBSWZFNRM-UHFFFAOYSA-N
Compound NameN-[2-[2-[[4-(3-tert-butyl-7-fluoro-2-methylbenzimidazol-5-yl)-5-fluoropyrimidin-2-yl]amino]-7,8-dihydro-5H-1,6-naphthyridin-6-yl]ethylidene]hydroxylamine
Canonical SMILESCc1nc2c(F)cc(-c3nc(Nc4ccc5c(n4)CCN(CC=NO)C5)ncc3F)cc2n1C(C)(C)C
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.43
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11802 CDK4 Homo sapiens Human PF00069 8.8 IC50 ChEMBL;BindingDB
Q00534 CDK6 Homo sapiens Human PF00069 8.6 IC50 ChEMBL;BindingDB
P24941 CDK2 Homo sapiens Human PF00069 7.8 IC50 ChEMBL;BindingDB