Molecule Details
InChIKeyOOOKPENMJKOYJM-UHFFFAOYSA-N
Compound Name6-(4-fluorophenyl)-5-[4-(quinolin-2-ylmethoxy)phenyl]-1H-pyridin-2-one
Canonical SMILESO=c1ccc(-c2ccc(OCc3ccc4ccccc4n3)cc2)c(-c2ccc(F)cc2)[nH]1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL8.11
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9Y233 PDE10A Homo sapiens Human PF01590 PF00233 8.8 IC50 ChEMBL;BindingDB
P41595 HTR2B Homo sapiens Human PF00001 7.4 IC50 ChEMBL;BindingDB