Molecule Details
InChIKeyOONYUIKMLKLQPP-GOSISDBHSA-N
Compound Name(R)-7-(4-fluorophenyl)-8-(1-methyl-1H-benzo[d] imidazol-6-yl)-2-((l-methylpyrrolidin-2-yl)meth yl)-[l,2,4]triazolo[1,5-c]pyrimidin-5-amine
Canonical SMILESCN1CCC[C@@H]1Cc1nc2c(-c3ccc4ncn(C)c4c3)c(-c3ccc(F)cc3)nc(N)n2n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.23
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P29274 ADORA2A Homo sapiens Human PF00001 9.0 IC50 ChEMBL;BindingDB
P30542 ADORA1 Homo sapiens Human PF00001 7.5 IC50 ChEMBL;BindingDB