Molecule Details
InChIKeyOOLJOHRMOKSYKO-QPJJXVBHSA-N
Compound Name4-(2-(5-cyano-4-(4-methyl-1H-indol-5-ylamino)pyridin-3-yl)vinyl)-N,N-dimethylbenzenesulfonamide
Canonical SMILESCc1c(Nc2c(C#N)cncc2/C=C/c2ccc(S(=O)(=O)N(C)C)cc2)ccc2[nH]ccc12
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL7.96
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P18505 GABRB1 Homo sapiens Human PF02931 PF02932 8.0 pIC50 TTD_MultiTarget
Q04759 PRKCQ Homo sapiens Human PF00130 PF21494 PF00069 PF00433 8.0 IC50 ChEMBL;BindingDB