Molecule Details
InChIKeyOOEHNCVFPNJDTF-UHFFFAOYSA-N
Canonical SMILESO=C(O)c1cccc(Cn2c(-c3ccc(Cl)cc3)nn(Cc3nnc(Cc4c(Cl)cccc4Cl)[nH]3)c2=O)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.38
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P30518 AVPR2 Homo sapiens Human PF00001 8.7 IC50 ChEMBL;BindingDB
P37288 AVPR1A Homo sapiens Human PF00001 PF08983 8.1 IC50 ChEMBL;BindingDB