Molecule Details
InChIKeyONYFRVQMWFWRSZ-HNNXBMFYSA-N
Compound Name5-[1-[6-[(3S)-3-aminopiperidin-1-yl]-2-pyridinyl]pyrazolo[4,3-c]pyridin-6-yl]-3-methylpyrazin-2-amine
Canonical SMILESCc1nc(-c2cc3c(cn2)cnn3-c2cccc(N3CCC[C@H](N)C3)n2)cnc1N
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL10.18
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q86V86 PIM3 Homo sapiens Human PF00069 11.0 Ki ChEMBL;BindingDB
P11309 PIM1 Homo sapiens Human PF00069 10.3 Ki ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 9.2 Ki ChEMBL;BindingDB