Molecule Details
InChIKeyOMXJXAHPPQYWRS-OGCSMFTJSA-N
Compound Name(1R,8R,9S,13S)-11-[2-(2-methoxyphenyl)prop-2-enoyl]-1-(4-methylphenyl)-11-azatetracyclo[6.5.2.0^{2,7}.0^{9,13}]pentadeca-2,4,6-triene-9-carboxylic acid
Canonical SMILESC=C(C(=O)N1C[C@H]2[C@@]3(c4ccc(C)cc4)CC[C@H](c4ccccc43)[C@@]2(C(=O)O)C1)c1ccccc1OC
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL8.1
SourceChEMBL;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P49354 FNTA Homo sapiens Human PF01239 8.1 pIC50 TTD_MultiTarget
P49356 FNTB Homo sapiens Human PF00432 8.1 IC50 ChEMBL