Molecule Details
InChIKeyOMSSRUBSGSKAFS-IPIAHOSKSA-N
Compound NameAc-Nle-c[Asp-Pro-Pro-D-Nal(2')-Arg-Trp-Lys]-NH2
Canonical SMILESCCCC[C@H](NC(C)=O)C(=O)N[C@H]1CC(=O)NCCCC[C@@H](C(N)=O)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](Cc2ccc3ccccc3c2)NC(=O)[C@@H]2CCCN2C(=O)[C@@H]2CCCN2C1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.29
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P41968 MC3R Homo sapiens Human PF00001 8.6 IC50 ChEMBL;BindingDB
P32245 MC4R Homo sapiens Human PF00001 6.7 IC50 ChEMBL;BindingDB
P33032 MC5R Homo sapiens Human PF00001 6.5 IC50 ChEMBL;BindingDB