Molecule Details
InChIKeyOMGQIHJJEYTELG-UHFFFAOYSA-N
Compound Name3-amino-6-[4-(2-methoxyethylsulfamoyl)phenyl]-N-pyridin-3-ylpyrazine-2-carboxamide
Canonical SMILESCOCCNS(=O)(=O)c1ccc(-c2cnc(N)c(C(=O)Nc3cccnc3)n2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)4
Pfam Stratification Cross-Family
Avg pChEMBL7.45
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (4)
Target Gene Organism Category Pfam pChEMBL Type Source
P49841 GSK3B Homo sapiens Human PF00069 8.7 Ki ChEMBL;BindingDB
O96020 CCNE2 Homo sapiens Human PF02984 PF00134 7.0 Ki ChEMBL
P24864 CCNE1 Homo sapiens Human PF02984 PF00134 7.0 Ki ChEMBL
P24941 CDK2 Homo sapiens Human PF00069 7.0 Ki ChEMBL