Molecule Details
InChIKeyOLZQDHRXJOXCLL-UHFFFAOYSA-N
Compound NameN-[5-cyano-4-(2-methoxyethoxy)-2-pyridinyl]-7-formyl-6-[1-(2,2,2-trifluoroethyl)piperidin-4-yl]-3,4-dihydro-2H-1,8-naphthyridine-1-carboxamide
Canonical SMILESCOCCOc1cc(NC(=O)N2CCCc3cc(C4CCN(CC(F)(F)F)CC4)c(C=O)nc32)ncc1C#N
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL7.61
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P22455 FGFR4 Homo sapiens Human PF07679 PF13927 PF07714 8.9 IC50 ChEMBL;BindingDB
Q12809 KCNH2 Homo sapiens Human PF00027 PF00520 PF13426 6.3 IC50 ChEMBL;BindingDB