Molecule Details
InChIKeyOLYGYSAFCXIBIB-UHFFFAOYSA-N
Compound Name8-N-cyclopentyl-2-N-(1-methylsulfonylpiperidin-4-yl)pyrido[3,4-d]pyrimidine-2,8-diamine
Canonical SMILESCS(=O)(=O)N1CCC(Nc2ncc3ccnc(NC4CCCC4)c3n2)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL9.07
SourceBindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P24941 CDK2 Homo sapiens Human PF00069 9.6 IC50 BindingDB
P24385 CCND1 Homo sapiens Human PF02984 PF00134 8.8 IC50 BindingDB
P11802 CDK4 Homo sapiens Human PF00069 8.8 IC50 BindingDB