Molecule Details
InChIKeyOLKXVDKTEYJKPA-UHFFFAOYSA-N
Compound NameN-methyl-5-[3-[6-(4-methylimidazol-1-yl)-2-pyridinyl]-1H-indol-5-yl]-1,3,4-thiadiazol-2-amine
Canonical SMILESCNc1nnc(-c2ccc3[nH]cc(-c4cccc(-n5cnc(C)c5)n4)c3c2)s1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.26
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q86V86 PIM3 Homo sapiens Human PF00069 8.8 IC50 ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 8.1 IC50 ChEMBL;BindingDB
P11309 PIM1 Homo sapiens Human PF00069 7.9 IC50 ChEMBL;BindingDB