Molecule Details
InChIKeyOLHTYSHHUSHAPW-UHFFFAOYSA-N
Compound Name2-{4-[4-(3-Trifluoromethylphenyl)piperazin-1-yl]butyl}amino-4-phenylpyridine
Canonical SMILESFC(F)(F)c1cccc(N2CCN(CCCCNc3cc(-c4ccccc4)ccn3)CC2)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.58
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P14416 DRD2 Homo sapiens Human PF00001 9.1 Ki ChEMBL;BindingDB
P35348 ADRA1A Homo sapiens Human PF00001 6.9 Ki ChEMBL;BindingDB
P35462 DRD3 Homo sapiens Human PF00001 6.7 Ki ChEMBL;BindingDB