Molecule Details
InChIKeyOLFPBASVCZUWSQ-UHFFFAOYSA-N
Compound Name7-methoxy-2-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)-2,3,4,5-tetrahydro-1H-benzo[c]azepin-1-one
Canonical SMILESCOc1ccc2c(c1)CCCN(CCCCN1CCN(c3ccccc3OC)CC1)C2=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.95
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P35462 DRD3 Homo sapiens Human PF00001 9.6 Ki ChEMBL;BindingDB
P14416 DRD2 Homo sapiens Human PF00001 8.8 Ki ChEMBL;BindingDB
P21917 DRD4 Homo sapiens Human PF00001 8.5 Ki ChEMBL