Molecule Details
InChIKeyOLCWFLWEHWLBTO-HSZRJFAPSA-N
Compound NameBms-214662
Canonical SMILESN#Cc1ccc2c(c1)CN(S(=O)(=O)c1cccs1)[C@H](Cc1ccccc1)CN2Cc1c[nH]cn1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)4
Pfam Stratification Cross-Family
Avg pChEMBL8.75
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
DrugBank Annotations
DrugBank ID DB12234
Drug NameBMS-214662
CAS Number195987-41-8
Groups investigational
ATC Codes nan
DescriptionBMS-214662 has been used in trials studying the treatment of Childhood Myelodysplastic Syndromes, Refractory Anemia With Excess Blasts, Recurrent Adult Acute Myeloid Leukemia, Relapsing Chronic Myelogenous Leukemia, and Adult Acute Promyelocytic Leukemia (M3), among others.

Categories: Benzazepines Heterocyclic Compounds, Fused-Ring
Cross-references: BindingDB: 50092365 CHEMBL351706 ChemSpider: 395310 PDB: BMV PubChem:448545 PubChem:347828513 ZINC: ZINC000003925649
Target Activities (4)
Target Gene Organism Category Pfam pChEMBL Type Source
P49354 FNTA Homo sapiens Human PF01239 9.2 pIC50 TTD_MultiTarget
P01112 HRAS Homo sapiens Human PF00071 8.9 IC50 ChEMBL
P49356 FNTB Homo sapiens Human PF00432 8.9 IC50 ChEMBL;BindingDB
P01116 KRAS Homo sapiens Human PF00071 8.1 IC50 ChEMBL
DrugBank Target Actions (2)
Target Gene Target Name Action Type
P49354 FNTA Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha modulator targets
P49356 FNTB Protein farnesyltransferase subunit beta modulator targets