Molecule Details
InChIKeyOKUPZBPYLVKVSU-UHFFFAOYSA-N
Compound Name2-{3-[3-(piperidin-4-yl)propoxy]phenyl}-N-[4-(1H-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]acetamide
Canonical SMILESO=C(Cc1cccc(OCCCC2CCNCC2)c1)Nc1nc(-c2c[nH]c3ncccc23)cs1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.8
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q13464 ROCK1 Homo sapiens Human PF25346 PF00069 PF08912 8.3 Ki ChEMBL;BindingDB
P36888 FLT3 Homo sapiens Human PF00047 PF07714 6.1 Ki ChEMBL;BindingDB
O75582 RPS6KA5 Homo sapiens Human PF00069 PF00433 6.0 Ki ChEMBL;BindingDB