Molecule Details
InChIKeyOKIZRSLVLMFZQA-UHFFFAOYSA-N
Compound Name2-[4-(2,6-Dioxo-1-propyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-phenoxy]-N-(2-hydroxy-ethyl)-acetamide
Canonical SMILESCCCn1c(=O)[nH]c2[nH]c(-c3ccc(OCC(=O)NCCO)cc3)nc2c1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.49
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P29275 ADORA2B Homo sapiens Human PF00001 8.9 Ki ChEMBL;BindingDB
P30542 ADORA1 Homo sapiens Human PF00001 7.2 Ki ChEMBL;BindingDB
P0DMS8 ADORA3 Homo sapiens Human PF00001 6.4 Ki ChEMBL;BindingDB