Molecule Details
InChIKeyOKIVGPUCUWMOIH-UHFFFAOYSA-N
Compound Name2-(4-Chloro-phenoxy)-N-[4-methyl-2-(4-methyl-piperazin-1-yl)-quinolin-6-yl]-acetamide
Canonical SMILESCc1cc(N2CCN(C)CC2)nc2ccc(NC(=O)COc3ccc(Cl)cc3)cc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.57
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q99705 MCHR1 Homo sapiens Human PF00001 7.2 IC50 ChEMBL;BindingDB
P41595 HTR2B Homo sapiens Human PF00001 6.5 IC50 ChEMBL;BindingDB
P28335 HTR2C Homo sapiens Human PF00001 6.0 IC50 ChEMBL;BindingDB