Molecule Details
InChIKeyOKAYCQSOIKKHMZ-KOZAUXTDSA-N
Compound Name6-Cyclohexylamino-9-((2R,3R,4S,5S)-3,4,5-trihydroxy-tetrahydro-furan-2-yl)-9H-purine-2-carbonitrile
Canonical SMILESN#Cc1nc(NC2CCCCC2)c2ncn([C@@H]3O[C@H](O)[C@@H](O)[C@H]3O)c2n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.95
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P43235 CTSK Homo sapiens Human PF08246 PF00112 8.0 IC50 ChEMBL;BindingDB
P25774 CTSS Homo sapiens Human PF08246 PF00112 6.5 IC50 ChEMBL;BindingDB
P07711 CTSL Homo sapiens Human PF08246 PF00112 6.4 IC50 ChEMBL;BindingDB