Molecule Details
InChIKeyOJQQCSPYLMDJQP-UHFFFAOYSA-N
Compound Name1-[3-Tert-butyl-1-[4-(2-morpholin-4-ylethoxy)phenyl]pyrazol-5-yl]-3-[4-[2-[(3-oxo-1,2-dihydroisoindol-5-yl)amino]pyrimidin-4-yl]oxynaphthalen-1-yl]urea
Canonical SMILESCC(C)(C)c1cc(NC(=O)Nc2ccc(Oc3ccnc(Nc4ccc5c(c4)C(=O)NC5)n3)c3ccccc23)n(-c2ccc(OCCN3CCOCC3)cc2)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.53
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P43405 SYK Homo sapiens Human PF07714 PF00017 8.0 IC50 ChEMBL;BindingDB
Q16539 MAPK14 Homo sapiens Human PF00069 7.8 IC50 ChEMBL;BindingDB
P49840 GSK3A Homo sapiens Human PF00069 6.7 IC50 ChEMBL;BindingDB