Molecule Details
InChIKeyOJODISRNMRYALN-UHFFFAOYSA-N
Compound Name1-(7-Carbamimidoyl-naphthalen-2-ylmethyl)-6-[1-(1-imino-ethyl)-piperidin-4-yloxy]-1H-indole-2-carboxylic acid methyl ester
Canonical SMILESCOC(=O)c1cc2ccc(OC3CCN(C(C)=N)CC3)cc2n1Cc1ccc2ccc(C(=N)N)cc2c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.75
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00742 F10 Homo sapiens Human PF00008 PF14670 PF00594 PF00089 9.7 Ki ChEMBL;BindingDB
P07477 PRSS1 Homo sapiens Human PF00089 6.8 Ki ChEMBL;BindingDB
P00734 F2 Homo sapiens Human PF00594 PF00051 PF09396 PF00089 6.7 Ki ChEMBL;BindingDB