Molecule Details
InChIKeyOIUQFNNWKMANNS-UHFFFAOYSA-N
Compound Name4-{1-[3-(Pyridin-2-ylamino)-phenyl]-3-pyrrolidin-1-yl-propylamino}-quinazoline-8-carboxylic acid amide
Canonical SMILESNC(=O)c1cccc2c(NC(CCN3CCCC3)c3cccc(Nc4ccccn4)c3)ncnc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.34
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q96GD4 AURKB Homo sapiens Human PF00069 8.3 IC50 ChEMBL;BindingDB
O14965 AURKA Homo sapiens Human PF00069 7.5 IC50 ChEMBL;BindingDB
P23443 RPS6KB1 Homo sapiens Human PF00069 PF00433 6.2 IC50 ChEMBL;BindingDB