Molecule Details
InChIKeyOITZRVNFLKKVDS-ODUWWZQZSA-N
Compound Name2-[(5S,10S,13S,17S)-17-[di(propan-2-yl)carbamoyl]-10,13-dimethyl-4,5,6,7,8,9,11,12,14,15,16,17-dodecahydro-1H-cyclopenta[a]phenanthren-3-yl]acetic acid
Canonical SMILESCC(C)N(C(=O)[C@H]1CCC2C3CC[C@H]4CC(CC(=O)O)=CC[C@]4(C)C3CC[C@@]21C)C(C)C
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL7.4
SourceTTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P18505 GABRB1 Homo sapiens Human PF02931 PF02932 7.4 pIC50 TTD_MultiTarget
P31639 SLC5A2 Homo sapiens Human PF00474 7.4 pIC50 TTD_MultiTarget