Molecule Details
InChIKeyOIQWAEIGTZYWRX-IGKWTDBASA-N
Canonical SMILESCC(C)(C)[C@H]1CC[C@H](N(Cc2ccc(C(=O)NC[C@H](O)C(=O)O)cc2)C(=O)Nc2cc(C(F)(F)F)cc(C(F)(F)F)c2)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.76
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P47871 GCGR Homo sapiens Human PF00002 PF02793 7.1 IC50 ChEMBL;BindingDB
P48546 GIPR Homo sapiens Human PF00002 PF02793 6.4 IC50 ChEMBL;BindingDB