Molecule Details
InChIKeyOILPCJZAWDBHHE-UHFFFAOYSA-N
Compound NameN-(3-Bromo-2''-sulfamoyl-biphenyl-4-yl)-2-(5-carbamimidoyl-1H-indol-3-yl)-acetamide
Canonical SMILESN=C(N)c1ccc2[nH]cc(CC(=O)Nc3ccc(-c4ccccc4S(N)(=O)=O)cc3Br)c2c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.7
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00742 F10 Homo sapiens Human PF00008 PF14670 PF00594 PF00089 9.5 Ki ChEMBL;BindingDB
P07477 PRSS1 Homo sapiens Human PF00089 6.9 Ki ChEMBL;BindingDB
P00734 F2 Homo sapiens Human PF00594 PF00051 PF09396 PF00089 6.7 Ki ChEMBL;BindingDB