Molecule Details
InChIKeyOHSIGBOKYLDSHG-RSXGOPAZSA-N
Compound NameN-(4-((((1S,2S)-2-(5-Fluoro-2-methoxyphenyl)cyclopropyl)methyl)(propyl)amino)butyl)-4-(pyridin-2-yl)benzamide
Canonical SMILESCCCN(CCCCNC(=O)c1ccc(-c2ccccn2)cc1)C[C@H]1C[C@@H]1c1cc(F)ccc1OC
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.95
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P35462 DRD3 Homo sapiens Human PF00001 8.1 Ki ChEMBL;BindingDB
P28335 HTR2C Homo sapiens Human PF00001 6.7 IC50 ChEMBL;BindingDB
P21917 DRD4 Homo sapiens Human PF00001 6.1 Ki ChEMBL;BindingDB