Molecule Details
InChIKeyOHIFKDNMHSXJFA-XAOJMSMDSA-N
Compound Name(3R)-7-hydroxy-N-[(2S)-1-[(3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl]-3-methylbutan-2-yl]-2-methyl-3,4-dihydro-1H-isoquinoline-3-carboxamide
Canonical SMILESCC(C)[C@@H](CN1CC[C@@](C)(c2cccc(O)c2)[C@@H](C)C1)NC(=O)[C@H]1Cc2ccc(O)cc2CN1C
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.04
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P41145 OPRK1 Homo sapiens Human PF00001 9.4 Ki ChEMBL;BindingDB
P35372 OPRM1 Homo sapiens Human PF00001 7.8 Ki ChEMBL;BindingDB
P41143 OPRD1 Homo sapiens Human PF00001 6.9 Ki ChEMBL;BindingDB