Molecule Details
InChIKeyOHENHOGCMRSJBB-QMMMGPOBSA-N
Compound Name4-[4-[(2S)-2-aminopropyl]sulfonyl-3-sulfamoyl-2-(2H-tetrazol-5-yl)phenyl]-1H-benzimidazole-2-carboxylic acid
Canonical SMILESC[C@H](N)CS(=O)(=O)c1ccc(-c2cccc3[nH]c(C(=O)O)nc23)c(-c2nn[nH]n2)c1S(N)(=O)=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL9.76
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
C7C422 blaNDM-1 Klebsiella pneumoniae Pathogen PF00753 10.1 IC50 ChEMBL;BindingDB
Q9XAY4 blaVIM Pseudomonas aeruginosa Pathogen PF00753 9.7 IC50 BindingDB
P52699 Serratia marcescens Pathogen PF00753 9.5 IC50 BindingDB