Molecule Details
InChIKeyOGZXGYFYZZWWML-UHFFFAOYSA-N
Compound Name2-Butyl-3-[[4-[2-[(2-cyclohexylacetyl)sulfamoyl]phenyl]phenyl]methyl]-5-(difluoromethylsulfanyl)imidazole-4-carboxylic acid
Canonical SMILESCCCCc1nc(SC(F)F)c(C(=O)O)n1Cc1ccc(-c2ccccc2S(=O)(=O)NC(=O)CC2CCCCC2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.6
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P30556 AGTR1 Homo sapiens Human PF00001 8.6 IC50 ChEMBL;BindingDB
P50052 AGTR2 Homo sapiens Human PF00001 8.6 IC50 ChEMBL