Molecule Details
InChIKeyOGNOHOPSWWOASA-UHFFFAOYSA-N
Compound Name4-[3-[3-(benzylsulfonylamino)-2,6-difluorobenzoyl]-2H-pyrazolo[3,4-b]pyridin-5-yl]benzenesulfonamide
Canonical SMILESNS(=O)(=O)c1ccc(-c2cnc3[nH]nc(C(=O)c4c(F)ccc(NS(=O)(=O)Cc5ccccc5)c4F)c3c2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.62
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P45985 MAP2K4 Homo sapiens Human PF00069 6.8 IC50 ChEMBL;BindingDB
P45983 MAPK8 Homo sapiens Human PF00069 6.7 Kd ChEMBL;BindingDB
P15056 BRAF Homo sapiens Human PF00130 PF07714 PF02196 6.3 Kd ChEMBL;BindingDB