Molecule Details
InChIKeyOGILCXDJHLQZTN-UHFFFAOYSA-N
Compound Name6-[[5-Amino-7-(4-fluorophenyl)-8-[imidazo[1,2-a] pyridin-6-yl]-[1,2,4]triazolo[1,5-c]pyrimidin-2-yl] methyl]pyridin-2-amine
Canonical SMILESNc1cccc(Cc2nc3c(-c4ccc5nccn5c4)c(-c4ccc(F)cc4)nc(N)n3n2)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.17
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P30542 ADORA1 Homo sapiens Human PF00001 8.4 IC50 ChEMBL;BindingDB
P29274 ADORA2A Homo sapiens Human PF00001 8.2 IC50 ChEMBL;BindingDB
P29275 ADORA2B Homo sapiens Human PF00001 7.9 IC50 ChEMBL;BindingDB