Molecule Details
InChIKeyOFDAQIKHAJYTBV-MRXNPFEDSA-N
Compound Name2-[3-(2-Fluoro-phenylmethanesulfonylamino)-2-oxo-2H-pyridin-1-yl]-N-((R)-1-formyl-4-guanidino-butyl)-acetamide
Canonical SMILESN=C(N)NCCC[C@@H](NC(=O)Cn1cccc(NS(=O)(=O)Cc2ccccc2F)c1=O)C(=O)O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.88
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00734 F2 Homo sapiens Human PF00594 PF00051 PF09396 PF00089 9.2 Ki ChEMBL;BindingDB
P07477 PRSS1 Homo sapiens Human PF00089 7.7 Ki ChEMBL;BindingDB
P00742 F10 Homo sapiens Human PF00008 PF14670 PF00594 PF00089 6.7 Ki ChEMBL;BindingDB