Molecule Details
InChIKeyOEYHDFBDGFEAHO-UHFFFAOYSA-N
Compound Name7-[1-(4,5,6,7-Tetrahydro-1-benzothiophene-2-carbonyl)piperidin-3-yl]-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonitrile
Canonical SMILESN#Cc1cc(C2CCCN(C(=O)c3cc4c(s3)CCCC4)C2)n2ncnc2n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.08
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
O00408 PDE2A Homo sapiens Human PF01590 PF00233 8.0 IC50 ChEMBL;BindingDB
Q13370 PDE3B Homo sapiens Human PF00233 6.2 IC50 ChEMBL;BindingDB