Molecule Details
InChIKeyOEYDBWKMXFZENQ-UHFFFAOYSA-N
Compound Name4-[(4-Chlorophenyl)methyl]-2-(1-methylazepan-3-yl)phthalazin-1-one
Canonical SMILESCN1CCCCC(n2nc(Cc3ccc(Cl)cc3)c3ccccc3c2=O)C1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.4
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P35367 HRH1 Homo sapiens Human PF00001 8.6 Ki ChEMBL;BindingDB
P35348 ADRA1A Homo sapiens Human PF00001 6.8 pIC50 TTD_MultiTarget
P35368 ADRA1B Homo sapiens Human PF00001 6.8 Ki ChEMBL