Molecule Details
InChIKeyOEXTZXWPZXNIIH-UHFFFAOYSA-N
Compound NameUS10428063, Example 14
Canonical SMILESCC(=O)Nc1cc(-c2[nH]c3c(c2Nc2ccccc2)C(=O)NCC3)ccn1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.47
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O43683 BUB1 Homo sapiens Human PF08311 PF00069 7.7 IC50 ChEMBL;BindingDB
P48729 CSNK1A1 Homo sapiens Human PF00069 7.7 IC50 BindingDB
P00533 EGFR Homo sapiens Human PF00757 PF14843 PF07714 PF01030 PF21314 7.0 IC50 BindingDB